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Dried Leaf Artemisia Annua Improves Bioavailability of Artemisinin via Cytochrome P450 Inhibition and Enhances Artemisinin Efficacy Downstream

Artemisia annua L. and artemisinin, have been used for millennia to treat malaria. We used human liver microsomes (HLM) and rats to compare hepatic metabolism, tissue distribution, and inflammation attenuation by dried leaves of A. annua (DLA) and pure artemisinin. For HLM assays, extracts, teas, an...

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Bibliografiske detaljer
Udgivet i:Biomolecules
Main Authors: Desrosiers, Matthew R., Mittleman, Alexis, Weathers, Pamela J.
Format: Artigo
Sprog:Inglês
Udgivet: MDPI 2020
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7072484/
https://ncbi.nlm.nih.gov/pubmed/32046156
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom10020254
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