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Dried Leaf Artemisia Annua Improves Bioavailability of Artemisinin via Cytochrome P450 Inhibition and Enhances Artemisinin Efficacy Downstream

Artemisia annua L. and artemisinin, have been used for millennia to treat malaria. We used human liver microsomes (HLM) and rats to compare hepatic metabolism, tissue distribution, and inflammation attenuation by dried leaves of A. annua (DLA) and pure artemisinin. For HLM assays, extracts, teas, an...

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Detalhes bibliográficos
Publicado no:Biomolecules
Main Authors: Desrosiers, Matthew R., Mittleman, Alexis, Weathers, Pamela J.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7072484/
https://ncbi.nlm.nih.gov/pubmed/32046156
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom10020254
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