Caricamento...

Targeting Receptor Tyrosine Kinase VEGFR-2 in Hepatocellular Cancer: Rational Design, Synthesis and Biological Evaluation of 1,2-Disubstituted Benzimidazoles

In this study, a novel series of 1,2-disubstituted benzo[d]imidazoles was rationally designed as VEGFR-2 inhibitors targeting hepatocellular carcinoma. Our design strategy is two-fold; it aimed first at studying the effect of replacing the 5-methylfuryl moiety of the well-known antiangiogenic 2-fury...

Descrizione completa

Salvato in:
Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Abdel-Mohsen, Heba T., Abdullaziz, Mona A., El Kerdawy, Ahmed M., Ragab, Fatma A. F., Flanagan, Keith J., Mahmoud, Abeer E. E., Ali, Mamdouh M., El Diwani, Hoda I., Senge, Mathias O.
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7071059/
https://ncbi.nlm.nih.gov/pubmed/32053964
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25040770
Tags: Aggiungi Tag
Nessun Tag, puoi essere il primo ad aggiungerne! !