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Aurantiamide-related dipeptide derivatives are formyl peptide receptor 1 antagonists

Formyl peptide receptor 1 (FPR1) is expressed on a variety of immune system cells and is a key regulator of the inflammatory environment. Therefore, the development of FPR1 antagonists may represent a novel approach for modulating innate immunity and treating inflammatory diseases. Starting from a d...

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Publicado en:Medchemcomm
Autores principales: Mastromarino, Margherita, Kirpotina, Liliya N., Schepetkin, Igor A., Quinn, Mark T., Lacivita, Enza, Leopoldo, Marcello
Formato: Artigo
Lenguaje:Inglês
Publicado: Royal Society of Chemistry 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7069519/
https://ncbi.nlm.nih.gov/pubmed/32206242
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c9md00336c
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