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Chemoselective Tertiary C—H Hydroxylation for Late-Stage Functionalization with Mn(PDP)/Chloroacetic Acid Catalysis

Aromatic and heterocyclic functionality are ubiquitous in pharmaceuticals. Herein, we disclose a new Mn(PDP)catalyst system using chloroacetic acid additive capable of chemoselectively oxidizing remote tertiary C(sp(3))—H bonds in the presence of a broad range of aromatic and heterocyclic moieties....

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Adv Synth Catal
Prif Awduron: Chambers, Rachel K., Zhao, Jinpeng, Delaney, Connor P., White, M. Christina
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2019
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC7066868/
https://ncbi.nlm.nih.gov/pubmed/32165875
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/adsc.201901472
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