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Effects of Strong CYP2C8 or CYP3A Inhibition and CYP3A Induction on the Pharmacokinetics of Brigatinib, an Oral Anaplastic Lymphoma Kinase Inhibitor, in Healthy Volunteers

In vitro data support involvement of cytochrome P450 (CYP)2C8 and CYP3A4 in the metabolism of the anaplastic lymphoma kinase inhibitor brigatinib. A 3‐arm, open‐label, randomized, single‐dose, fixed‐sequence crossover study was conducted to characterize the effects of the strong inhibitors gemfibroz...

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Detalhes bibliográficos
Publicado no:Clin Pharmacol Drug Dev
Main Authors: Tugnait, Meera, Gupta, Neeraj, Hanley, Michael J., Sonnichsen, Daryl, Kerstein, David, Dorer, David J., Venkatakrishnan, Karthik, Narasimhan, Narayana
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7027746/
https://ncbi.nlm.nih.gov/pubmed/31287236
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cpdd.723
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