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Lysosomal Fusion: An Efficient Mechanism Increasing Their Sequestration Capacity for Weak Base Drugs without Apparent Lysosomal Biogenesis

Lysosomal sequestration of anticancer therapeutics lowers their cytotoxic potential, reduces drug availability at target sites, and contributes to cancer resistance. Only recently has it been shown that lysosomal sequestration of weak base drugs induces lysosomal biogenesis mediated by activation of...

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Pubblicato in:Biomolecules
Autori principali: Skoupa, Nikola, Dolezel, Petr, Mlejnek, Petr
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7022710/
https://ncbi.nlm.nih.gov/pubmed/31947839
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom10010077
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