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Structure guided prediction of Pyrazinamide resistance mutations in pncA

Pyrazinamide plays an important role in tuberculosis treatment; however, its use is complicated by side-effects and challenges with reliable drug susceptibility testing. Resistance to pyrazinamide is largely driven by mutations in pyrazinamidase (pncA), responsible for drug activation, but genetic h...

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Detalhes bibliográficos
Publicado no:Sci Rep
Main Authors: Karmakar, Malancha, Rodrigues, Carlos H. M., Horan, Kristy, Denholm, Justin T., Ascher, David B.
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group UK 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7002382/
https://ncbi.nlm.nih.gov/pubmed/32024884
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-020-58635-x
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