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Synthesis and biological evaluation of [(11)C]SB366791: A new PET-radioligand for in vivo imaging of the TRPV1 receptor

INTRODUCTION: The transient receptor potential vanilloid subfamily member 1 (TRPV1) receptor, a non-selective cation channel, is known for its key role in pain nociception and neurogenic inflammation. TRPV1 expression has been demonstrated in diverse tissues and an essential role for TRPV1 in variou...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Nucl Med Biol
Prif Awduron: van Veghel, Daisy, Cleynhens, Jan, Pearce, Larry V., Blumberg, Peter M., Van Laere, Koen, Verbruggen, Alfons, Bormans, Guy
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2012
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6959540/
https://ncbi.nlm.nih.gov/pubmed/23141549
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2012.08.011
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