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Structural Dynamics Behind Clinical Mutants of PncA-Asp12Ala, Pro54Leu, and His57Pro of Mycobacterium tuberculosis Associated With Pyrazinamide Resistance

Pyrazinamide (PZA) is one of the main FDA approved drugs to be used as the first line of defense against Mycobacterium Tuberculosis (MTB). It is activated into pyrazinoic acid (POA) via MTB's pncA gene-encoded pyrazinamidase (PZase). Mutations are most commonly responsible for PZA-resistance in...

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Detalhes bibliográficos
Publicado no:Front Bioeng Biotechnol
Main Authors: Mehmood, Aamir, Khan, Muhammad Tahir, Kaushik, Aman Chandra, Khan, Anwar Sheed, Irfan, Muhammad, Wei, Dong-Qing
Formato: Artigo
Idioma:Inglês
Publicado em: Frontiers Media S.A. 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6914729/
https://ncbi.nlm.nih.gov/pubmed/31921809
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fbioe.2019.00404
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