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Combined in silico and (19)F NMR analysis of 5-fluorouracil metabolism in yeast at low ATP conditions

The cytotoxic effect of 5-fluorouracil (5-FU) on yeast cells is thought to be mainly via a misincorporation of fluoropyrimidines into both RNA and DNA, not only DNA damage via inhibition of thymidylate synthase (TYMS) by fluorodeoxyuridine monophosphate (FdUMP). However, some studies on Saccharomyce...

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Shranjeno v:
Bibliografske podrobnosti
izdano v:Biosci Rep
Main Authors: Pawłowski, Piotr H., Szczęsny, Paweł, Rempoła, Bożenna, Poznańska, Anna, Poznański, Jarosław
Format: Artigo
Jezik:Inglês
Izdano: Portland Press Ltd. 2019
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6904775/
https://ncbi.nlm.nih.gov/pubmed/31742586
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BSR20192847
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