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Insights into the Interaction Mechanisms of the Proviral Integration Site of Moloney Murine Leukemia Virus (Pim) Kinases with Pan-Pim Inhibitors PIM447 and AZD1208: A Molecular Dynamics Simulation and MM/GBSA Calculation Study

Based on the up-regulation of the proviral integration site of the Moloney murine leukemia virus (Pim) kinase family (Pim1, 2, and 3) observed in several types of leukemias and lymphomas, the development of pan-Pim inhibitors is an attractive therapeutic strategy. While only PIM447 and AZD1208 have...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Chen, Qingqing, Wang, Yan, Shi, Shanshan, Li, Kaihang, Zhang, Ling, Gao, Jian
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6862308/
https://ncbi.nlm.nih.gov/pubmed/31671637
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20215410
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