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Dasatinib Inhibits Procoagulant and Clot Retracting Activities of Human Platelets

Tyrosine kinase inhibitors (TKI) such as the BCR-ABL inhibitor dasatinib and nilotinib are highly effective therapies for chronic myeloid leukemia (CML). However, several lines of evidence suggest that dasatinib can induce bleeding which may be due to impaired collagen-induced platelet adhesion, agg...

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Опубликовано в: :Int J Mol Sci
Главные авторы: Beke Debreceni, Ildikó, Mezei, Gabriella, Batár, Péter, Illés, Árpád, Kappelmayer, János
Формат: Artigo
Язык:Inglês
Опубликовано: MDPI 2019
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6862041/
https://ncbi.nlm.nih.gov/pubmed/31683623
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20215430
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