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Dasatinib Inhibits Procoagulant and Clot Retracting Activities of Human Platelets

Tyrosine kinase inhibitors (TKI) such as the BCR-ABL inhibitor dasatinib and nilotinib are highly effective therapies for chronic myeloid leukemia (CML). However, several lines of evidence suggest that dasatinib can induce bleeding which may be due to impaired collagen-induced platelet adhesion, agg...

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Détails bibliographiques
Publié dans:Int J Mol Sci
Auteurs principaux: Beke Debreceni, Ildikó, Mezei, Gabriella, Batár, Péter, Illés, Árpád, Kappelmayer, János
Format: Artigo
Langue:Inglês
Publié: MDPI 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6862041/
https://ncbi.nlm.nih.gov/pubmed/31683623
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20215430
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