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Neurovascular drug biotransformation machinery in focal human epilepsies: Brain CYP3A4 correlates with seizure frequency and antiepileptic drug therapy

Pharmacoresistance is a major clinical challenge for approximately 30% of patients with epilepsy. Previous studies indicate nuclear receptors (NRs), efflux transporters and cytochrome P450 enzymes (CYPs) control drug passage across the blood-brain barrier (BBB) in drug resistant epilepsy. Here we 1)...

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Dades bibliogràfiques
Publicat a:Mol Neurobiol
Autors principals: Williams, Sherice, Hossain, Mohammed, Ferguson, Lisa, Busch, Robyn M., Marchi, Nicola, Gonzalez-Martinez, Jorge, Perucca, Emilio, Najm, Imad M., Ghosh, Chaitali
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6854685/
https://ncbi.nlm.nih.gov/pubmed/31243719
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s12035-019-01673-y
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