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The role of water and protein flexibility in the structure-based virtual screening of allosteric GPCR modulators: an mGlu(5) receptor case study

Stabilizing unique receptor conformations, allosteric modulators of G-protein coupled receptors (GPCRs) might open novel treatment options due to their new pharmacological action, their enhanced specificity and selectivity in both binding and signaling. Ligand binding occurs at intrahelical alloster...

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Bibliografische gegevens
Gepubliceerd in:J Comput Aided Mol Des
Hoofdauteurs: Orgován, Zoltán, Ferenczy, György G., Keserű, György M.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: Springer International Publishing 2019
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6825653/
https://ncbi.nlm.nih.gov/pubmed/31542869
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-019-00224-w
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