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The role of water and protein flexibility in the structure-based virtual screening of allosteric GPCR modulators: an mGlu(5) receptor case study

Stabilizing unique receptor conformations, allosteric modulators of G-protein coupled receptors (GPCRs) might open novel treatment options due to their new pharmacological action, their enhanced specificity and selectivity in both binding and signaling. Ligand binding occurs at intrahelical alloster...

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Bibliografiske detaljer
Udgivet i:J Comput Aided Mol Des
Main Authors: Orgován, Zoltán, Ferenczy, György G., Keserű, György M.
Format: Artigo
Sprog:Inglês
Udgivet: Springer International Publishing 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6825653/
https://ncbi.nlm.nih.gov/pubmed/31542869
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-019-00224-w
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