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The role of water and protein flexibility in the structure-based virtual screening of allosteric GPCR modulators: an mGlu(5) receptor case study

Stabilizing unique receptor conformations, allosteric modulators of G-protein coupled receptors (GPCRs) might open novel treatment options due to their new pharmacological action, their enhanced specificity and selectivity in both binding and signaling. Ligand binding occurs at intrahelical alloster...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:J Comput Aided Mol Des
Egile Nagusiak: Orgován, Zoltán, Ferenczy, György G., Keserű, György M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Springer International Publishing 2019
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6825653/
https://ncbi.nlm.nih.gov/pubmed/31542869
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-019-00224-w
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