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Curcumin-Synthetic Analogs Library Screening by Docking and Quantitative Structure–Activity Relationship Studies for AXL Tyrosine Kinase Inhibition in Cancers

AXL is an important drug target for cancers. Two-dimensional quantitative structure–activity relationship (2D-QSAR) tests were performed to elucidate a relationship between molecular structures and the activity of a series of 400 curcumin derivatives subjected to AXL kinase by ATP competition in the...

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Publicat a:J Comput Biol
Autors principals: Ghrifi, Fatima, Allam, Loubna, Wiame, Lakhlili, Ibrahimi, Azeddine
Format: Artigo
Idioma:Inglês
Publicat: Mary Ann Liebert, Inc., publishers 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6786334/
https://ncbi.nlm.nih.gov/pubmed/31009237
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1089/cmb.2019.0052
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