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Allosteric Control of Gating and Kinetics at P2X(4)Receptor Channels

The CNS abundantly expresses P2X receptor channels for ATP; of these the most widespread in the brain is the P2X(4)channel. We show that ivermectin (IVM) is a specific positive allosteric effector of heterologously expressed P2X(4) and possibly of heteromeric P2X(4)/P2X(6)channels, but not of P2X(2)...

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Bibliographic Details
Published in:J Neurosci
Main Authors: Khakh, Baljit S., Proctor, William R., Dunwiddie, Thomas V., Labarca, Cesar, Lester, Henry A.
Format: Artigo
Language:Inglês
Published: Society for Neuroscience 1999
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6782529/
https://ncbi.nlm.nih.gov/pubmed/10460235
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.19-17-07289.1999
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