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Distinct CRC-associated Apc mutations dictate response to Tankyrase inhibition

The majority of colorectal cancers (CRCs) show hyperactivated WNT signaling due to inactivating mutations in the APC tumor suppressor. Genetically restoring Apc suppresses WNT and induces rapid and sustained tumor regression, implying that re-engaging this endogenous tumor suppressive mechanism may...

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Dades bibliogràfiques
Publicat a:Cancer Discov
Autors principals: Schatoff, Emma M., Goswami, Sukanya, Zafra, Maria Paz, Foronda, Miguel, Shusterman, Michael, Leach, Benjamin I., Katti, Alyna, Diaz, Bianca J., Dow, Lukas E.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6774804/
https://ncbi.nlm.nih.gov/pubmed/31337618
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/2159-8290.CD-19-0289
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