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The Anticancer Agent Elesclomol Has Direct Effects on Mitochondrial Bioenergetic Function in Isolated Mammalian Mitochondria

Elesclomol ((N-malonyl-bis(N′-methyl-N′-thiobenzoylhydrazide)); formerly STA-4783) is a mitochondria-targeted chemotherapeutic agent that has demonstrated efficacy in selective cancer cell killing in pre-clinical and clinical testing. The biologically active form of elesclomol is a deprotonated copp...

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Detalhes bibliográficos
Publicado no:Biomolecules
Main Authors: Modica-Napolitano, Josephine S., Bharath, Leena P., Hanlon, Alison J., Hurley, Liam D.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6724019/
https://ncbi.nlm.nih.gov/pubmed/31344923
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom9080298
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