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First-In-Class Inhibitors Targeting the Interaction between Bacterial RNA Polymerase and Sigma Initiation Factor Affect the Viability and Toxin Release of Streptococcus pneumoniae

Novel antimicrobial classes are in desperate need for clinical management of infections caused by increasingly prevalent multi-drug resistant pathogens. The protein-protein interaction between bacterial RNA polymerase (RNAP) and the housekeeping sigma initiation factor is essential to transcription...

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Pubblicato in:Molecules
Autori principali: Ye, Jiqing, Chu, Adrian Jun, Lin, Lin, Yang, Xiao, Ma, Cong
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6719014/
https://ncbi.nlm.nih.gov/pubmed/31405060
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24162902
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