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Repurposing Quinacrine against Ebola Virus Infection In Vivo

Quinacrine hydrochloride is a small-molecule, orally bioavailable drug that has been used clinically as an antimalarial and for many other applications. A machine learning model trained on Ebola virus (EBOV) screening data identified quinacrine as a potent (nanomolar) in vitro inhibitor. In the curr...

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Dades bibliogràfiques
Publicat a:Antimicrob Agents Chemother
Autors principals: Lane, Thomas R., Comer, Jason E., Freiberg, Alexander N., Madrid, Peter B., Ekins, Sean
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6709481/
https://ncbi.nlm.nih.gov/pubmed/31307979
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01142-19
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