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One-Pot Synthesis of Benzo[4(,)5]imidazo[2(,)1-a]isoquinolines and Isoquinolino[3(,)4-b]quinoxalines via Tandem Cyclization Strategies

Two operationally simple one-pot protocols have been developed for the synthesis of amino-functionalized benzo[4,5]imidazo[2,1–a]isoquinolines and isoquinolino[3,4–b]quinoxalines. Optimization data and substrate scope for these atom-economical transformations, which engage commercially available o-p...

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Detalhes bibliográficos
Publicado no:J Org Chem
Main Authors: Bagdasarian, Alex L., Nguyen, Huy H., Palazzo, Teresa A., Fettinger, James C., Haddadin, Makhluf J., Kurth, Mark J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6688609/
https://ncbi.nlm.nih.gov/pubmed/27030441
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.joc.6b00338
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