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3-(4-Chloro-2-Morpholin-4-yl-Thiazol-5-yl)-8-(1-Ethylpropyl)-2,6-Dimethyl-Imidazo[1,2-b]Pyridazine: A Novel Brain-Penetrant, Orally Available Corticotropin-Releasing Factor Receptor 1 Antagonist with Efficacy in Animal Models of Alcoholism

We describe a novel corticotropin-releasing factor receptor 1 (CRF(1)) antagonist with advantageous properties for clinical development, and its in vivo activity in preclinical alcoholism models. 3-(4-Chloro-2-morpholin-4-yl-thiazol-5-yl)-8-(1-ethylpropyl)-2,6-dimethyl-imidazo[1,2-b]pyridazine (MTIP...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
में प्रकाशित:J Neurosci
मुख्य लेखकों: Gehlert, Donald R., Cippitelli, Andrea, Thorsell, Annika, Lê, Anh Dzung, Hipskind, Philip A., Hamdouchi, Chafiq, Lu, Jianliang, Hembre, Erik J., Cramer, Jeffrey, Song, Min, McKinzie, David, Morin, Michelle, Ciccocioppo, Roberto, Heilig, Markus
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: Society for Neuroscience 2007
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC6672492/
https://ncbi.nlm.nih.gov/pubmed/17344409
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.4985-06.2007
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