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Synthesis of pyrrolo[1,2-a]quinolines by formal 1,3-dipolar cycloaddition reactions of quinolinium salts

Quinolinium salts, Q(+)-CH(2)-CO(2)Me Br(−) and Q(+)-CH(2)-CONMe(2) Br(−) (where Q = quinoline), were prepared from quinolines. Deprotonation of these salts with triethylamine promoted the reaction of the resulting quinolinium ylides (formally azomethine ylides) with electron-poor alkenes by conjuga...

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Publicat a:Beilstein J Org Chem
Autors principals: Choi, Anthony, Morley, Rebecca M, Coldham, Iain
Format: Artigo
Idioma:Inglês
Publicat: Beilstein-Institut 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6633155/
https://ncbi.nlm.nih.gov/pubmed/31354865
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.15.149
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