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Influence of Obesity and Type 2 Diabetes Mellitus on the Pharmacokinetics of Tramadol After Single Oral Dose Administration

BACKGROUND AND OBJECTIVES: The number of overweight, obese and diabetic patients is constantly increasing. Metabolic disorders may affect the pharmacokinetics of drugs, e.g., by altering the activity of cytochrome P450 (CYP) isoenzymes. Tramadol is a commonly used analgesic metabolised mainly via CY...

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Detalhes bibliográficos
Publicado no:Eur J Drug Metab Pharmacokinet
Main Authors: Porażka, Joanna, Szałek, Edyta, Połom, Wojciech, Czajkowski, Mateusz, Grabowski, Tomasz, Matuszewski, Marcin, Grześkowiak, Edmund
Formato: Artigo
Idioma:Inglês
Publicado em: Springer International Publishing 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6616205/
https://ncbi.nlm.nih.gov/pubmed/30778911
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s13318-019-00543-1
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