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Computational methods and tools to predict cytochrome P450 metabolism for drug discovery

In this review, we present important, recent developments in the computational prediction of cytochrome P450 (CYP) metabolism in the context of drug discovery. We discuss in silico models for the various aspects of CYP metabolism prediction, including CYP substrate and inhibitor predictors, site of...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Chem Biol Drug Des
Egile Nagusiak: Tyzack, Jonathan D., Kirchmair, Johannes
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: John Wiley and Sons Inc. 2019
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6590657/
https://ncbi.nlm.nih.gov/pubmed/30471192
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cbdd.13445
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