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Omega-conotoxin GVIA binding to a high-affinity receptor in brain: characterization, calcium sensitivity, and solubilization

We describe unique, high-affinity binding sites for omega[125I]conotoxin GVIA in membranes from rat brain and rabbit sympathetic ganglia which appear to be primarily associated with N-type voltage-dependent calcium channels. The dissociation constant (KD) for the toxin in rat brain membranes is 60 p...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:J Neurosci
Prif Awduron: Wagner, JA, Snowman, AM, Biswas, A, Olivera, BM, Snyder, SH
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: Society for Neuroscience 1988
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6569423/
https://ncbi.nlm.nih.gov/pubmed/2845019
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.08-09-03354.1988
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