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The binding of kappa- and sigma-opiates in rat brain

Detailed displacements of [3H]dihydromorphine by ketocyclazocine and SKF 10,047, [3H]ethylketocyclazocine by SKF 10,047, and [3H]SKF 10,047 by ketocyclazocine are all multiphasic, suggesting multiple binding sites. After treating brain tissue in vitro with naloxazone, all displacements lose the init...

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Pubblicato in:J Neurosci
Autori principali: Wolozin, BL, Nishimura, S, Pasternak, GW
Natura: Artigo
Lingua:Inglês
Pubblicazione: Society for Neuroscience 1982
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6564346/
https://ncbi.nlm.nih.gov/pubmed/6283040
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1523/JNEUROSCI.02-06-00708.1982
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