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Properties of Opiate-Receptor Binding in Rat Brain

[(3)H]Naloxone, a potent opiate antagonist, binds stereospecifically to opiate-receptor sites in rat-brain tissue. The binding is time, temperature, and pH dependent and saturable with respect to [(3)H]naloxone and tissue concentration. The [(3)H]naloxone-receptor complex formation is bimolecular wi...

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Autors principals: Pert, Candace B., Snyder, Solomon H.
Format: Artigo
Idioma:Inglês
Publicat: 1973
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC433710/
https://ncbi.nlm.nih.gov/pubmed/4525427
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