Properties of Opiate-Receptor Binding in Rat Brain
[(3)H]Naloxone, a potent opiate antagonist, binds stereospecifically to opiate-receptor sites in rat-brain tissue. The binding is time, temperature, and pH dependent and saturable with respect to [(3)H]naloxone and tissue concentration. The [(3)H]naloxone-receptor complex formation is bimolecular wi...
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| Publicado en: | Proc Natl Acad Sci U S A |
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| Principais autores: | , |
| Formato: | Artigo |
| Idioma: | Inglês |
| Publicado: |
National Academy of Sciences
1973
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| Assuntos: | |
| Acceso en liña: | https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC433710/ https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/4525427/ https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.70.8.2243 |
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