Yüklüyor......

Fluorescent indomethacin-dansyl conjugates utilize the membrane-binding domain of cyclooxygenase-2 to block the opening to the active site

Many indomethacin amides and esters are cyclooxygenase-2 (COX-2)–selective inhibitors, providing a framework for the design of COX-2–targeted imaging and cancer chemotherapeutic agents. Although previous studies have suggested that the amide or ester moiety of these inhibitors binds in the lobby reg...

Ful tanımlama

Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:J Biol Chem
Asıl Yazarlar: Uddin, Md. Jashim, Banerjee, Surajit, Duggan, Kelsey, Musee, Joel, Kiefer, James R., Ghebreselasie, Kebreab, Rouzer, Carol A., Marnett, Lawrence J.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Society for Biochemistry and Molecular Biology 2019
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6552414/
https://ncbi.nlm.nih.gov/pubmed/31000626
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA119.007405
Etiketler: Etiketle
Etiket eklenmemiş, İlk siz ekleyin!