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Enhancement of Binding Affinity of Folate to Its Receptor by Peptide Conjugation

(1) Background: The folate receptor (FR) is a target for cancer treatment and detection. Expression of the FR is restricted in normal cells but overexpressed in many types of tumors. Folate was conjugated with peptides for enhancing binding affinity to the FR. (2) Materials and Methods: For conjugat...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Dharmatti, Roopa, Miyatake, Hideyuki, Nandakumar, Avanashiappan, Ueda, Motoki, Kobayashi, Kenya, Kiga, Daisuke, Yamamura, Masayuki, Ito, Yoshihiro
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6539678/
https://ncbi.nlm.nih.gov/pubmed/31052315
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20092152
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