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Wild-Type IDH Enzymes as Actionable Targets for Cancer Therapy

Isocitrate dehydrogenases (IDHs) are enzymes that catalyze the oxidative decarboxylation of isocitrate, producing α-ketoglutarate (αKG) and CO(2). The discovery of IDH1 and IDH2 mutations in several malignancies has brought to the approval of drugs targeting IDH1/2 mutants in cancers. Here, we summa...

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Detalhes bibliográficos
Publicado no:Cancers (Basel)
Main Authors: Bergaggio, Elisa, Piva, Roberto
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6520797/
https://ncbi.nlm.nih.gov/pubmed/31010244
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cancers11040563
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