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Development of Highly Selective 1,2,3-Triazole-containing Peptidic Polo-like Kinase 1 Polo-box Domain-binding Inhibitors

Members of the polo-like kinase (Plk) family of serine/threonine protein kinases play crucial roles in cell cycle regulation and proliferation. Of the five Plks (Plk1–5), Plk1 is recognized as an anticancer drug target. Plk1 contains multiple structural components that are important for its proper b...

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Publicat a:Molecules
Autors principals: Zhao, Xue Zhi, Tsuji, Kohei, Hymel, David, Burke, Terrence R.
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2019
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6515314/
https://ncbi.nlm.nih.gov/pubmed/31014020
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules24081488
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