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Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation

[Image: see text] A series of (E)-3-(4-((2,4-bis(trifluoromethyl)benzyl)oxy)-3-methoxyphenyl)-2-cyanoacrylamide derivatives were designed and synthesized as new estrogen-related receptor α (ERRα) degraders based on the proteolysis targeting chimera (PROTAC) concept. One of the representative compoun...

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Pubblicato in:ACS Med Chem Lett
Autori principali: Peng, Lijie, Zhang, Zhensheng, Lei, Chong, Li, Shan, Zhang, Zhang, Ren, Xiaomei, Chang, Yu, Zhang, Yan, Xu, Yong, Ding, Ke
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2019
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6512006/
https://ncbi.nlm.nih.gov/pubmed/31097997
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00025
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