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Biased TAS2R Bronchodilators Inhibit Airway Smooth Muscle Growth by Downregulating Phosphorylated Extracellular Signal–regulated Kinase 1/2

Bitter taste receptor (TAS2R) agonists dilate airways by receptor-dependent smooth muscle relaxation. Besides their coupling to relaxation, we have found that human airway smooth muscle (HASM) cell TAS2Rs activate (phosphorylate) extracellular signal–related kinase 1/2 (ERK1/2), but the cellular eff...

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Опубликовано в: :Am J Respir Cell Mol Biol
Главные авторы: Kim, Donghwa, Cho, Soomin, Castaño, Maria A., Panettieri, Reynold A., Woo, Jung A., Liggett, Stephen B.
Формат: Artigo
Язык:Inglês
Опубликовано: American Thoracic Society 2019
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6503617/
https://ncbi.nlm.nih.gov/pubmed/30365340
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1165/rcmb.2018-0189OC
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