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Synthesis and discovery of asiatic acid based 1,2,3-triazole derivatives as antitumor agents blocking NF-κB activation and cell migration

A series of asiatic acid (AA) based 1,2,3-triazole derivatives were designed, synthesized and subjected to a cell-based NF-κB inhibition screening assay. Among the tested compounds, compound 6k displayed impressive NF-κB inhibitory activity with an IC(50) value in the low micromolar range. A molecul...

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Bibliografiske detaljer
Udgivet i:Medchemcomm
Main Authors: Huang, Ri-Zhen, Liang, Gui-Bin, Li, Mei-Shan, Fang, Yi-Lin, Zhao, Shi-Feng, Zhou, Mei-Mei, Liao, Zhi-Xin, Sun, Jing, Wang, Heng-Shan
Format: Artigo
Sprog:Inglês
Udgivet: Royal Society of Chemistry 2019
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Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6484948/
https://ncbi.nlm.nih.gov/pubmed/31057738
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8md00620b
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