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Mechanistic Assessment of Extrahepatic Contributions to Glucuronidation of Integrase Strand Transfer Inhibitors

Integrase strand transfer inhibitor (INSTI)–based regimens dominate initial human immunodeficiency virus treatment. Most INSTIs are metabolized predominantly via UDP-glucuronosyltransferases (UGTs). For drugs predominantly metabolized by UGTs, including INSTIs, in vitro data recovered from human liv...

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Bibliographische Detailangaben
Veröffentlicht in:Drug Metab Dispos
Hauptverfasser: Liu, Stephanie N., Lu, Jessica Bo Li, Watson, Christy J. W., Lazarus, Philip, Desta, Zeruesenay, Gufford, Brandon T.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The American Society for Pharmacology and Experimental Therapeutics 2019
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6474910/
https://ncbi.nlm.nih.gov/pubmed/30804050
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.118.085035
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