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Investigation of Crystallization and Salt Formation of Poorly Water-Soluble Telmisartan for Enhanced Solubility

The crystal changes and salt formation of poorly water-soluble telmisartan (TEL) in various solvents were investigated for enhanced solubility, stability and crystallinity. Polymorphic behaviors of TEL were characterized by dispersing in distilled water, acetone, acetonitrile, DMSO, or ethanol using...

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Dettagli Bibliografici
Pubblicato in:Pharmaceutics
Autori principali: Park, Chulhun, Meghani, Nileshkumar M., Shin, Yongkwan, Oh, Euichaul, Park, Jun-Bom, Cui, Jing-Hao, Cao, Qing-Ri, Tran, Thao Truong-Dinh, Tran, Phuong Ha-Lien, Lee, Beom-Jin
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6470926/
https://ncbi.nlm.nih.gov/pubmed/30823389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics11030102
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