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2-Nitroimidazole-Furanoside Derivatives for Hypoxia Imaging—Investigation of Nucleoside Transporter Interaction, (18)F-Labeling and Preclinical PET Imaging

The benefits of PET imaging of tumor hypoxia in patient management has been demonstrated in many examples and with various tracers over the last years. Although, the optimal hypoxia imaging agent has yet to be found, 2-nitroimidazole (azomycin) sugar derivatives—mimicking nucleosides—have proven the...

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Publicat a:Pharmaceuticals (Basel)
Autors principals: Maier, Florian C., Schweifer, Anna, Damaraju, Vijaya L., Cass, Carol E., Bowden, Gregory D., Ehrlichmann, Walter, Kneilling, Manfred, Pichler, Bernd J., Hammerschmidt, Friedrich, Reischl, Gerald
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6469291/
https://ncbi.nlm.nih.gov/pubmed/30781409
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph12010031
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