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On-Resin Macrocyclization of Peptides Using Vinyl Sulfonamides as a Thiol-Michael “Click” Acceptor

Macrocyclization of linear peptides imparts improved stability to enzymatic degradation and increases potency of function. Many successful macrocyclization of peptides both in solution and on-resin have been achieved but are limited in scope as they lack selectivity, require long reaction times, or...

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Vydáno v:Bioconjug Chem
Hlavní autoři: Sutherland, Bryan P., El-Zaatari, Bassil M., Halaszynski, Nicole I., French, Jonathan M., Bai, Shi, Kloxin, Christopher J.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6467758/
https://ncbi.nlm.nih.gov/pubmed/30452234
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.bioconjchem.8b00751
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