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Targeted Inhibition of Plasmodium falciparum Calcium-Dependent Protein Kinase 1 with a Constrained J Domain-Derived Disruptor Peptide

To explore the possibility of constrained peptides to target Plasmodium-infected cells, we designed a J domain mimetic derived from Plasmodium falciparum calcium-dependent protein kinase 1 (Pf CDPK1) as a strategy to disrupt J domain binding and inhibit Pf CDPK1 activity. The J domain disruptor (JDD...

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Detalhes bibliográficos
Publicado no:ACS Infect Dis
Main Authors: Flaherty, Briana R., Ho, Tienhuei G., Schmidt, Sven H., Herberg, Friedrich W., Peterson, David S., Kennedy, Eileen J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6461495/
https://ncbi.nlm.nih.gov/pubmed/30746930
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.8b00347
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