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Potentiation of imatinib by cilostazol in sensitive and resistant gastrointestinal stromal tumor cell lines involves YAP inhibition

Despite the introduction of tyrosine kinase inhibitors, gastrointestinal stromal tumors (GIST) resistance remains a major clinical challenge. We previously identified phosphodiesterase 3A (PDE3A) as a potential therapeutic target expressed in most GIST. The PDE3 inhibitor cilostazol reduced cell via...

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Detalhes bibliográficos
Publicado no:Oncotarget
Main Authors: Vandenberghe, Pierre, Delvaux, Marine, Hagué, Perrine, Erneux, Christophe, Vanderwinden, Jean-Marie
Formato: Artigo
Idioma:Inglês
Publicado em: Impact Journals LLC 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6442998/
https://ncbi.nlm.nih.gov/pubmed/30956759
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.18632/oncotarget.26734
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