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Nitro Sulfonyl Fluorides are a new pharmacophore for the development of antibiotics

The development of antibiotics against Gram-negative bacteria is a central problem in drug discovery. In this report, we demonstrate that aromatic sulfonyl fluorides with a nitro group in their ortho position have remarkable antibacterial activity and are active against drug-resistant pathogens, suc...

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Dettagli Bibliografici
Pubblicato in:Mol Syst Des Eng
Autori principali: Sadlowski, Corinne, Park, Bora, Araújo, Clarissa, Das, Subhamoy, Kerr, D. Lucas, He, Maomao, Han, Hesong, Riley, Lee, Murthy, Niren
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6366622/
https://ncbi.nlm.nih.gov/pubmed/30740245
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C8ME00011E
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