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The importance of protonation and tautomerization in relative binding affinity prediction: a comparison of AMBER TI and Schrödinger FEP

In drug discovery, protonation states and tautomerization are easily overlooked. Through a Merck–Rutgers collaboration, this paper re-examined the initial settings and preparations for the Thermodynamic Integration (TI) calculation in AMBER Free-Energy Workflows, demonstrating the value of careful c...

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Bibliografiska uppgifter
I publikationen:J Comput Aided Mol Des
Huvudupphovsmän: Hu, Yuan, Sherborne, Brad, Lee, Tai-Sung, Case, David A., York, Darrin M., Guo, Zhuyan
Materialtyp: Artigo
Språk:Inglês
Publicerad: 2016
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC6360336/
https://ncbi.nlm.nih.gov/pubmed/27480697
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s10822-016-9920-5
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