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A New Approach for Improving the Antibacterial and Tumor Cytotoxic Activities of Pipemidic Acid by Including It in Trimethyl-β-cyclodextrin

Pipemidic acid (HPPA) is a quinolone antibacterial agent used mostly to treat gram-negative infections of the urinary tract, but its therapeutic use is limited because of its low solubility. Thus, to improve drug solubility, natural cyclodextrins (CDs) are used for their ability of including guest m...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Lavorgna, Margherita, Iacovino, Rosa, Russo, Chiara, Di Donato, Cristina, Piscitelli, Concetta, Isidori, Marina
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6359225/
https://ncbi.nlm.nih.gov/pubmed/30669399
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20020416
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