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Discovery of a 3,4,5-trisubstituted-1,2,4-triazole agonist with high affinity and selectivity at the somatostatin subtype-4 (sst(4)) receptor

A series of compounds containing a 1,2,4-triazole moiety were synthesized, targeting the somatostatin receptor subtype-4 (sst(4)). Compounds were developed in which the Phe(6)/Phe(7)/Phe(11), Trp(8), and Lys(9) mimetic groups were interchanged at positions 3, 4, and 5 of the 1,2,4-triazole ring. The...

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Bibliografiske detaljer
Udgivet i:Medchemcomm
Main Authors: Daryaei, Iman, Sandoval, Karin, Witt, Ken, Kontoyianni, Maria, Michael Crider, A.
Format: Artigo
Sprog:Inglês
Udgivet: Royal Society of Chemistry 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6336083/
https://ncbi.nlm.nih.gov/pubmed/30746066
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8md00388b
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